manual_drip
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Caffeine Analogs
Many are stronger then caffeine (1,3-Dipropyl 7-Proparagyl Xanthine is 100 times stronger). Many have stronger effects on A2 then A1 adenosine receptors compared to caffeine. I heard once that antagonizes one of the adenosine receptors caused restlessness and antagonizing the other one caused more desireable stimulation - anyone know which is which? If A2 is better the more selective analogs would likely have cleaner effects than caffeine.
Many are stronger then caffeine (1,3-Dipropyl 7-Proparagyl Xanthine is 100 times stronger). Many have stronger effects on A2 then A1 adenosine receptors compared to caffeine. I heard once that antagonizes one of the adenosine receptors caused restlessness and antagonizing the other one caused more desireable stimulation - anyone know which is which? If A2 is better the more selective analogs would likely have cleaner effects than caffeine.